Compile Data Set for Download or QSAR
maximum 50k data
Found 31 of ic50 data for polymerid = 1246
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557849(1-(3-((4-((3,4-dichlorophenyl)amino)-7-methoxyquin...)
Affinity DataIC50:  3.20nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557865(1-(4-((4-((3,4-dichloro- phenyl)amino)-7-methoxy- ...)
Affinity DataIC50:  6.5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557852(1-(3-((4-((3,4-dichloro-2-fluorophenyl)amino)-7-me...)
Affinity DataIC50:  9.5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557872(1-(4-((4-((4-bromo-3- chlorophenyl)amino)-7- metho...)
Affinity DataIC50:  11nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557851(1-(3-((4-((2,4-dichlorophenyl)amino)-7-methoxyquin...)
Affinity DataIC50:  14nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557868(1-(3-((4-((4-bromo-3- chlorophenyl)amino)-7- metho...)
Affinity DataIC50:  17nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557875(1-(3-((7-methoxy-4- (phenylamino)quinazolin-6- yl)...)
Affinity DataIC50:  18nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557857(6-((1-acryloylpiperidin-4- yl)oxy)-4-((2,4-dichlor...)
Affinity DataIC50:  20nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557870(1-(3-((4-((3,4-dichloro-2- fluorophenyl)amino)-7- ...)
Affinity DataIC50:  21nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557846(1-(4-((4-((2,4-dichlorophenyl)amino)-7-methoxyquin...)
Affinity DataIC50:  21nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557850(6-((1-acryloylpiperidin-4-yl)oxy)-4-((3,4-dichloro...)
Affinity DataIC50:  25nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557873(1-(4-((7-methoxy-4- (phenylamino)quinazolin-6- yl)...)
Affinity DataIC50:  50nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557854(US11365189, Ex. No. 9)
Affinity DataIC50:  79nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557869(1-(3-((4-((3-cyclopropyl- phenyl)amino)-7-methoxy-...)
Affinity DataIC50:  79nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557853(6-((1-acryloylpiperidin-4-yl)oxy)-4-((3,4-dichloro...)
Affinity DataIC50:  100nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557871(1-(3-((7-methoxy-4-((4- (trifluoromethyl)phenyl)- ...)
Affinity DataIC50:  110nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557876(1-(3-((4-((3-chloro-4- (trifluoromethoxy)phenyl)- ...)
Affinity DataIC50:  150nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557867(1-(4-((7-methoxy-4-((3- (oxazol-5-yl)phenyl)- amin...)
Affinity DataIC50:  200nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557856(6-((1-acryloylpiperidin-4- yl)oxy)-4-((3-(hydroxy-...)
Affinity DataIC50:  260nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557881(1-(3-((4-((4-bromo-3- chlorophenyl)amino)- pyrido[...)
Affinity DataIC50:  270nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557860(6-((1-acryloylpiperidin-4- yl)oxy)-4-((4-chloro-3-...)
Affinity DataIC50:  300nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557880(1-(3-((4-((4-chloro-3- (hydroxymethyl)phenyl)- ami...)
Affinity DataIC50:  300nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557877(1-(3-((7-methoxy-4-((3- (oxazol-5-yl)phenyl)- amin...)
Affinity DataIC50:  320nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557878(1-(3-((7-methoxy-4- (phenylamino)quinazolin-6- yl)...)
Affinity DataIC50:  350nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557874(1-(3-((4-((2,4-dichloro- phenyl)amino)-7-methoxy- ...)
Affinity DataIC50:  510nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557866(1-(3-((7-methoxy-4-((3- (oxazol-5-yl)phenyl)- amin...)
Affinity DataIC50:  710nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557848(1-(3-((4-((2,4-dichlorophenyl)amino)pyrido[3,4-d]p...)
Affinity DataIC50:  760nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557861(6-((1-acryloylpiperidin-4- yl)oxy)-7-methoxy-4-((3...)
Affinity DataIC50:  1.30E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557858(6-((1-acryloylpiperidin-4- yl)oxy)-4-((4-bromo-3- ...)
Affinity DataIC50:  3.20E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557855(6-((1-acryloylpiperidin-4- yl)oxy)-4-((4-chloro-3-...)
Affinity DataIC50:  8.90E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2 [1-780,'GSP',781-1255](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557879(1-(3-((7-methoxy-4-((1- methyl-1H-indazol-7-yl)- a...)
Affinity DataIC50:  9.10E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent